Ketoconazole inhibits the cellular uptake of anandamide via inhibition of FAAH at pharmacologically relevant concentrations.

Björklund, Emmelie

Ketoconazole inhibits the cellular uptake of anandamide via inhibition of FAAH at pharmacologically relevant concentrations. [electronic resource] - PloS one 2014 - e87542 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1932-6203

10.1371/journal.pone.0087542 doi


Amidohydrolases--antagonists & inhibitors
Analysis of Variance
Arachidonic Acids--metabolism
Caco-2 Cells
Dose-Response Relationship, Drug
Endocannabinoids--metabolism
Hep G2 Cells
Humans
Ketoconazole--pharmacology
Polyunsaturated Alkamides--metabolism
Receptor, Cannabinoid, CB2--metabolism