Structure-activity relationships and blood distribution of antiplasmodial aminopeptidase-1 inhibitors. [electronic resource]
Producer: 20130314Description: 10909-17 p. digitalISSN:- 1520-4804
- Aminopeptidases -- antagonists & inhibitors
- Animals
- Antimalarials -- blood
- Cell Line
- Drug Resistance
- Female
- Humans
- Malaria -- drug therapy
- Malonates -- blood
- Metalloproteases -- antagonists & inhibitors
- Mice
- Molecular Docking Simulation
- Plasmodium berghei
- Plasmodium falciparum -- drug effects
- Protein Binding
- Protozoan Proteins -- antagonists & inhibitors
- Rats
- Solubility
- Stereoisomerism
- Structure-Activity Relationship
- Tissue Distribution
- Zinc
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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