The feasibility of enzyme targeted activation for amino acid/dipeptide monoester prodrugs of floxuridine; cathepsin D as a potential targeted enzyme. [electronic resource]
Producer: 20120719Description: 3672-89 p. digitalISSN:- 1420-3049
- Amino Acids -- metabolism
- Antimetabolites, Antineoplastic -- metabolism
- Cathepsin B -- metabolism
- Cathepsin D -- metabolism
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Dipeptides -- metabolism
- Drug Stability
- Enzyme Activation -- drug effects
- Floxuridine -- metabolism
- Gene Expression Profiling
- Gene Expression Regulation, Neoplastic -- drug effects
- Humans
- Pancreatic Neoplasms -- drug therapy
- Prodrugs -- metabolism
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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