An in vitro Förster resonance energy transfer-based high-throughput screening assay for inhibitors of protein-protein interactions in SUMOylation pathway. [electronic resource]
Producer: 20121231Description: 336-43 p. digitalISSN:- 1557-8127
- Algorithms
- DNA -- genetics
- Dose-Response Relationship, Drug
- Escherichia coli -- drug effects
- Fluorescence Resonance Energy Transfer -- methods
- Fluorescent Antibody Technique
- Gene Expression -- drug effects
- High-Throughput Screening Assays -- methods
- Humans
- Metabolic Networks and Pathways -- drug effects
- Polymerase Chain Reaction
- Recombinant Fusion Proteins -- chemistry
- Reproducibility of Results
- SUMO-1 Protein -- metabolism
- Signal-To-Noise Ratio
- Sumoylation -- drug effects
- Ubiquitin-Conjugating Enzymes -- metabolism
- Urea -- pharmacology
- Ubiquitin-Conjugating Enzyme UBC9
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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