An in vitro Förster resonance energy transfer-based high-throughput screening assay for inhibitors of protein-protein interactions in SUMOylation pathway.
Song, Yang
An in vitro Förster resonance energy transfer-based high-throughput screening assay for inhibitors of protein-protein interactions in SUMOylation pathway. [electronic resource] - Assay and drug development technologies Aug 2012 - 336-43 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1557-8127
10.1089/adt.2011.0394 doi
Algorithms
DNA--genetics
Dose-Response Relationship, Drug
Escherichia coli--drug effects
Fluorescence Resonance Energy Transfer--methods
Fluorescent Antibody Technique
Gene Expression--drug effects
High-Throughput Screening Assays--methods
Humans
Metabolic Networks and Pathways--drug effects
Polymerase Chain Reaction
Recombinant Fusion Proteins--chemistry
Reproducibility of Results
SUMO-1 Protein--metabolism
Signal-To-Noise Ratio
Sumoylation--drug effects
Ubiquitin-Conjugating Enzymes--metabolism
Urea--pharmacology
Ubiquitin-Conjugating Enzyme UBC9
An in vitro Förster resonance energy transfer-based high-throughput screening assay for inhibitors of protein-protein interactions in SUMOylation pathway. [electronic resource] - Assay and drug development technologies Aug 2012 - 336-43 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1557-8127
10.1089/adt.2011.0394 doi
Algorithms
DNA--genetics
Dose-Response Relationship, Drug
Escherichia coli--drug effects
Fluorescence Resonance Energy Transfer--methods
Fluorescent Antibody Technique
Gene Expression--drug effects
High-Throughput Screening Assays--methods
Humans
Metabolic Networks and Pathways--drug effects
Polymerase Chain Reaction
Recombinant Fusion Proteins--chemistry
Reproducibility of Results
SUMO-1 Protein--metabolism
Signal-To-Noise Ratio
Sumoylation--drug effects
Ubiquitin-Conjugating Enzymes--metabolism
Urea--pharmacology
Ubiquitin-Conjugating Enzyme UBC9