Significant species difference in amide hydrolysis of GDC-0834, a novel potent and selective Bruton's tyrosine kinase inhibitor. [electronic resource]
Producer: 20120329Description: 1840-9 p. digitalISSN:- 1521-009X
- Agammaglobulinaemia Tyrosine Kinase
- Amides -- metabolism
- Animals
- Cells, Cultured
- Clinical Trials, Phase I as Topic
- Dogs
- Double-Blind Method
- Female
- Hepatocytes -- metabolism
- Humans
- Hydrolysis
- Macaca fascicularis
- Male
- Mice
- Microsomes, Liver -- metabolism
- Protein Kinase Inhibitors -- metabolism
- Protein-Tyrosine Kinases -- antagonists & inhibitors
- Pyrimidinones -- metabolism
- Randomized Controlled Trials as Topic
- Rats
- Rats, Sprague-Dawley
- Species Specificity
- Thiophenes -- metabolism
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Publication Type: Journal Article
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