Activity and the metabolic activation pathway of the potent and selective hepatitis C virus pronucleotide inhibitor PSI-353661. [electronic resource]
Producer: 20111109Description: 120-32 p. digitalISSN:- 1872-9096
- Antiviral Agents -- pharmacology
- Biotransformation
- Cathepsin A -- metabolism
- Chromatography, High Pressure Liquid
- Cloning, Molecular
- Drug Evaluation, Preclinical
- Guanosine Monophosphate -- analogs & derivatives
- Guanylate Kinases -- metabolism
- Hep G2 Cells
- Hepacivirus -- drug effects
- Hepatocytes -- drug effects
- Humans
- Lactic Acid -- metabolism
- Luciferases -- metabolism
- Microbial Sensitivity Tests
- Mitochondria -- drug effects
- Mutation
- Nerve Tissue Proteins -- metabolism
- Phenol -- metabolism
- Phosphorylation
- Prodrugs -- chemistry
- Replicon
- Viral Nonstructural Proteins -- antagonists & inhibitors
- Virus Replication -- drug effects
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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