Biological properties of androgen receptor pure antagonist for treatment of castration-resistant prostate cancer: optimization from lead compound to CH5137291. [electronic resource]
Producer: 20110926Description: 1344-56 p. digitalISSN:- 1097-0045
- Androgen Antagonists -- pharmacokinetics
- Androgen Receptor Antagonists -- administration & dosage
- Anilides -- pharmacokinetics
- Animals
- Antineoplastic Agents -- pharmacology
- Carbamates -- pharmacology
- Cell Nucleus -- metabolism
- Cell Proliferation -- drug effects
- Cells, Cultured
- Dose-Response Relationship, Drug
- Humans
- Lead
- Male
- Mice
- Mice, Nude
- Mice, SCID
- Neoplasm Transplantation
- Nitriles -- metabolism
- Orchiectomy
- Prostatic Neoplasms -- metabolism
- Receptors, Androgen -- drug effects
- Sulfonamides -- administration & dosage
- Thiohydantoins -- administration & dosage
- Tosyl Compounds -- pharmacokinetics
- Transcription, Genetic -- drug effects
- Translocation, Genetic
- Transplantation, Heterologous
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Publication Type: Comparative Study; Journal Article
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