Discovery of 1-(3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-2-imidazolidinone (GSK163090), a Potent, selective, and orally active 5-HT1A/B/D receptor antagonist. [electronic resource]
Producer: 20140415Description: 8228-40 p. digitalISSN:- 1520-4804
- Administration, Oral
- Animals
- CHO Cells
- Chromatography, Liquid
- Cricetulus
- Drug Discovery
- Humans
- Imidazoles -- administration & dosage
- Magnetic Resonance Spectroscopy
- Male
- Quinolines -- administration & dosage
- Rats, Sprague-Dawley
- Receptors, Serotonin -- classification
- Serotonin Antagonists -- administration & dosage
- Tandem Mass Spectrometry
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Publication Type: Journal Article
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