Mutations that increase both Hsp90 ATPase activity in vitro and Hsp90 drug resistance in vivo. [electronic resource]
Producer: 20100628Description: 575-83 p. digitalISSN:- 0006-3002
- Adenosine Triphosphatases -- metabolism
- Amino Acid Substitution
- Benzoquinones -- pharmacology
- Blotting, Western
- Chaperonins -- genetics
- Drug Resistance
- Enzyme Inhibitors -- pharmacology
- HSP90 Heat-Shock Proteins -- antagonists & inhibitors
- Humans
- Immunoprecipitation
- In Vitro Techniques
- Kidney -- embryology
- Lactams, Macrocyclic -- pharmacology
- Models, Molecular
- Molecular Chaperones -- genetics
- Mutation -- genetics
- Protein Binding
- Protein Conformation
- Saccharomyces cerevisiae -- genetics
- Saccharomyces cerevisiae Proteins -- genetics
- Two-Hybrid System Techniques
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Publication Type: Journal Article
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