Mutations that increase both Hsp90 ATPase activity in vitro and Hsp90 drug resistance in vivo.

Zurawska, Anna

Mutations that increase both Hsp90 ATPase activity in vitro and Hsp90 drug resistance in vivo. [electronic resource] - Biochimica et biophysica acta May 2010 - 575-83 p. digital

Publication Type: Journal Article

0006-3002

10.1016/j.bbamcr.2010.03.002 doi


Adenosine Triphosphatases--metabolism
Amino Acid Substitution
Benzoquinones--pharmacology
Blotting, Western
Chaperonins--genetics
Drug Resistance
Enzyme Inhibitors--pharmacology
HSP90 Heat-Shock Proteins--antagonists & inhibitors
Humans
Immunoprecipitation
In Vitro Techniques
Kidney--embryology
Lactams, Macrocyclic--pharmacology
Models, Molecular
Molecular Chaperones--genetics
Mutation--genetics
Protein Binding
Protein Conformation
Saccharomyces cerevisiae--genetics
Saccharomyces cerevisiae Proteins--genetics
Two-Hybrid System Techniques