C-5 Substituted heteroaryl 3-pyridinecarbonitriles as PKCtheta inhibitors: Part I. [electronic resource]
Producer: 20091123Description: 5423-5 p. digitalISSN:- 1464-3405
- Animals
- Inhibitory Concentration 50
- Isoenzymes -- antagonists & inhibitors
- Mice
- Mice, Knockout
- Nitriles -- chemistry
- Protein Kinase C -- antagonists & inhibitors
- Protein Kinase C-theta
- Protein Kinase Inhibitors -- chemistry
- Pyridines -- chemistry
- Structure-Activity Relationship
- T-Lymphocytes -- drug effects
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Publication Type: Journal Article
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