Small intestinal efflux mediated by MRP2 and BCRP shifts sulfasalazine intestinal permeability from high to low, enabling its colonic targeting. [electronic resource]
Producer: 20090825Description: G371-7 p. digitalISSN:- 1522-1547
- 2-Pyridinylmethylsulfinylbenzimidazoles -- pharmacology
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- metabolism
- ATP Binding Cassette Transporter, Subfamily G, Member 2
- ATP-Binding Cassette Transporters -- antagonists & inhibitors
- Administration, Oral
- Animals
- Biological Transport
- Caco-2 Cells
- Colon -- drug effects
- Dose-Response Relationship, Drug
- Drug Delivery Systems
- Humans
- Indoles -- pharmacology
- Indomethacin -- pharmacology
- Intestinal Absorption
- Intestine, Small -- drug effects
- Kinetics
- Male
- Multidrug Resistance-Associated Protein 2
- Multidrug Resistance-Associated Proteins -- antagonists & inhibitors
- Neoplasm Proteins -- antagonists & inhibitors
- Pantoprazole
- Perfusion
- Permeability
- Propionates -- pharmacology
- Quinolines -- pharmacology
- Rats
- Rats, Wistar
- Sulfasalazine -- administration & dosage
No physical items for this record
Publication Type: Journal Article
There are no comments on this title.
Log in to your account to post a comment.