The selective 5-hydroxytryptamine 1A antagonist, AZD7371 [3(R)-(N,N-dicyclobutylamino)-8-fluoro-3,4-dihydro-2H-1-benzopyran-5-carboxamide (R,R)-tartrate monohydrate] (robalzotan tartrate monohydrate), inhibits visceral pain-related visceromotor, but not autonomic cardiovascular, responses to colorectal distension in rats. [electronic resource]
Producer: 20090623Description: 1048-55 p. digitalISSN:- 1521-0103
- Abdominal Muscles -- drug effects
- Abdominal Pain -- drug therapy
- Animals
- Benzopyrans -- administration & dosage
- Blood Pressure -- drug effects
- Cardiovascular Physiological Phenomena -- drug effects
- Colonic Diseases -- complications
- Dilatation, Pathologic -- complications
- Disease Models, Animal
- Dose-Response Relationship, Drug
- Female
- Heart Rate -- drug effects
- Piperazines -- pharmacology
- Pyridines -- pharmacology
- Rats
- Rats, Sprague-Dawley
- Serotonin 5-HT1 Receptor Antagonists
- Serotonin Antagonists -- administration & dosage
- Urination -- drug effects
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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