Elucidating rifampin's inducing and inhibiting effects on glyburide pharmacokinetics and blood glucose in healthy volunteers: unmasking the differential effects of enzyme induction and transporter inhibition for a drug and its primary metabolite. [electronic resource]
Producer: 20090106Description: 78-85 p. digitalISSN:- 1532-6535
- Administration, Oral
- Adult
- Anti-Infective Agents -- pharmacology
- Area Under Curve
- Blood Glucose -- drug effects
- Ciprofloxacin -- pharmacology
- Drug Interactions
- Enzyme Induction -- drug effects
- Enzyme Inhibitors -- administration & dosage
- Female
- Glyburide -- metabolism
- Humans
- Hypoglycemic Agents -- metabolism
- Infusions, Intravenous
- Liver -- drug effects
- Liver-Specific Organic Anion Transporter 1 -- drug effects
- Male
- Metabolic Clearance Rate
- Rifampin -- administration & dosage
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Publication Type: Clinical Trial; Journal Article; Research Support, N.I.H., Extramural
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