Elucidating rifampin's inducing and inhibiting effects on glyburide pharmacokinetics and blood glucose in healthy volunteers: unmasking the differential effects of enzyme induction and transporter inhibition for a drug and its primary metabolite.

Zheng, H X

Elucidating rifampin's inducing and inhibiting effects on glyburide pharmacokinetics and blood glucose in healthy volunteers: unmasking the differential effects of enzyme induction and transporter inhibition for a drug and its primary metabolite. [electronic resource] - Clinical pharmacology and therapeutics Jan 2009 - 78-85 p. digital

Publication Type: Clinical Trial; Journal Article; Research Support, N.I.H., Extramural

1532-6535

10.1038/clpt.2008.186 doi


Administration, Oral
Adult
Anti-Infective Agents--pharmacology
Area Under Curve
Blood Glucose--drug effects
Ciprofloxacin--pharmacology
Drug Interactions
Enzyme Induction--drug effects
Enzyme Inhibitors--administration & dosage
Female
Glyburide--metabolism
Humans
Hypoglycemic Agents--metabolism
Infusions, Intravenous
Liver--drug effects
Liver-Specific Organic Anion Transporter 1--drug effects
Male
Metabolic Clearance Rate
Rifampin--administration & dosage