Identification, characterization and initial hit-to-lead optimization of a series of 4-arylamino-3-pyridinecarbonitrile as protein kinase C theta (PKCtheta) inhibitors. [electronic resource]
Producer: 20081030Description: 5958-63 p. digitalISSN:- 1520-4804
- Animals
- Crystallography, X-Ray
- Dose-Response Relationship, Drug
- Drug Evaluation, Preclinical
- Female
- Indoles -- chemical synthesis
- Interleukin-2 -- antagonists & inhibitors
- Isoenzymes -- antagonists & inhibitors
- Mice
- Mice, Inbred C57BL
- Mice, Knockout
- Models, Molecular
- Molecular Structure
- Nitriles -- chemical synthesis
- Protein Kinase C -- antagonists & inhibitors
- Protein Kinase C-theta
- Protein Kinase Inhibitors -- chemical synthesis
- Pyridines -- chemical synthesis
- Spleen -- cytology
- Stereoisomerism
- Structure-Activity Relationship
- T-Lymphocytes -- drug effects
No physical items for this record
Publication Type: Journal Article
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