TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists. [electronic resource]
Producer: 20071123Description: 815-7 p. digitalISSN:- 1095-9203
- 6-Cyano-7-nitroquinoxaline-2,3-dione -- chemistry
- Animals
- Benzodiazepines -- pharmacology
- Binding, Competitive
- Cell Line
- Cerebellum -- cytology
- Crystallography, X-Ray
- Drug Partial Agonism
- Hippocampus -- cytology
- Humans
- In Vitro Techniques
- Interneurons -- drug effects
- Mice
- Models, Molecular
- Patch-Clamp Techniques
- Protein Conformation
- Protein Subunits -- physiology
- Pyramidal Cells -- drug effects
- Quinoxalines -- pharmacology
- Receptors, AMPA -- agonists
- Structure-Activity Relationship
- Synaptic Transmission -- drug effects
- Trichlormethiazide -- pharmacology
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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