TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists.
Menuz, Karen
TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists. [electronic resource] - Science (New York, N.Y.) Nov 2007 - 815-7 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1095-9203
10.1126/science.1146317 doi
6-Cyano-7-nitroquinoxaline-2,3-dione--chemistry
Animals
Benzodiazepines--pharmacology
Binding, Competitive
Cell Line
Cerebellum--cytology
Crystallography, X-Ray
Drug Partial Agonism
Hippocampus--cytology
Humans
In Vitro Techniques
Interneurons--drug effects
Mice
Models, Molecular
Patch-Clamp Techniques
Protein Conformation
Protein Subunits--physiology
Pyramidal Cells--drug effects
Quinoxalines--pharmacology
Receptors, AMPA--agonists
Structure-Activity Relationship
Synaptic Transmission--drug effects
Trichlormethiazide--pharmacology
TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists. [electronic resource] - Science (New York, N.Y.) Nov 2007 - 815-7 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1095-9203
10.1126/science.1146317 doi
6-Cyano-7-nitroquinoxaline-2,3-dione--chemistry
Animals
Benzodiazepines--pharmacology
Binding, Competitive
Cell Line
Cerebellum--cytology
Crystallography, X-Ray
Drug Partial Agonism
Hippocampus--cytology
Humans
In Vitro Techniques
Interneurons--drug effects
Mice
Models, Molecular
Patch-Clamp Techniques
Protein Conformation
Protein Subunits--physiology
Pyramidal Cells--drug effects
Quinoxalines--pharmacology
Receptors, AMPA--agonists
Structure-Activity Relationship
Synaptic Transmission--drug effects
Trichlormethiazide--pharmacology