Discovery of N1-(6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonyl)tryptamine as a potent, selective, and orally active 5-HT(6) receptor agonist. [electronic resource]
Producer: 20080108Description: 5535-8 p. digitalISSN:- 0022-2623
- Administration, Oral
- Animals
- Biological Availability
- CHO Cells
- Cricetinae
- Cricetulus
- Dogs
- Frontal Lobe -- metabolism
- Haplorhini
- Humans
- In Vitro Techniques
- Mice
- Microdialysis
- Microsomes, Liver -- metabolism
- Radioligand Assay
- Rats
- Receptors, Serotonin -- metabolism
- Serotonin Receptor Agonists -- chemical synthesis
- Solubility
- Structure-Activity Relationship
- Thiazoles -- chemistry
- Tryptamines -- chemical synthesis
- gamma-Aminobutyric Acid -- metabolism
No physical items for this record
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
There are no comments on this title.
Log in to your account to post a comment.