The anxioselective agent 7-(2-chloropyridin-4-yl)pyrazolo-[1,5-a]-pyrimidin-3-yl](pyridin-2-yl)methanone (DOV 51892) is more efficacious than diazepam at enhancing GABA-gated currents at alpha1 subunit-containing GABAA receptors. [electronic resource]
Producer: 20070109Description: 1244-52 p. digitalISSN:- 0022-3565
- Animals
- Anti-Anxiety Agents -- chemical synthesis
- Ataxia -- chemically induced
- Chloride Channels -- drug effects
- Diazepam -- pharmacology
- Dose-Response Relationship, Drug
- Exploratory Behavior -- drug effects
- Hand Strength -- physiology
- Hypnotics and Sedatives -- pharmacology
- Male
- Motor Activity -- drug effects
- Muscle Relaxation -- drug effects
- Oocytes -- metabolism
- Postural Balance -- drug effects
- Pyrazoles -- chemical synthesis
- Pyridines -- chemical synthesis
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Rats, Wistar
- Receptors, GABA-A -- drug effects
- Xenopus laevis
- gamma-Aminobutyric Acid -- physiology
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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