Aripiprazole and its human metabolite are partial agonists at the human dopamine D2 receptor, but the rodent metabolite displays antagonist properties. [electronic resource]
Producer: 20070111Description: 88-94 p. digitalISSN:- 0014-2999
- Amphetamine
- Animals
- Antipsychotic Agents -- metabolism
- Aripiprazole
- Behavior, Animal -- drug effects
- Binding, Competitive
- Biotransformation
- CHO Cells
- Catalepsy -- chemically induced
- Cricetinae
- Cricetulus
- Dopamine D2 Receptor Antagonists
- Dyskinesia, Drug-Induced -- etiology
- Guanosine 5'-O-(3-Thiotriphosphate) -- metabolism
- HeLa Cells
- Humans
- Male
- Motor Activity -- drug effects
- Oxidopamine
- Piperazines -- metabolism
- Quinolones -- metabolism
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptors, Dopamine D2 -- agonists
- Species Specificity
- Transfection
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Publication Type: Comparative Study; Journal Article
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