Identification and initial evaluation of 4-N-aryl-[1,4]diazepane ureas as potent CXCR3 antagonists. [electronic resource]
Producer: 20060321Description: 200-3 p. digitalISSN:- 0960-894X
- Calcium -- metabolism
- Cell Line
- Chemistry, Pharmaceutical -- methods
- Chemokine CXCL11
- Chemokines, CXC -- chemistry
- Chemotaxis
- Dose-Response Relationship, Drug
- Drug Design
- Drug Evaluation, Preclinical
- Electrons
- Humans
- Inflammation
- Inhibitory Concentration 50
- Models, Chemical
- Receptors, CXCR3
- Receptors, Chemokine -- antagonists & inhibitors
- Receptors, G-Protein-Coupled -- metabolism
- Recombinant Proteins -- chemistry
- Stereoisomerism
- T-Lymphocytes -- cytology
- Urea -- chemistry
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Publication Type: Journal Article
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