2-Aminoethoxydiphenyl borate (2-APB) antagonises inositol 1,4,5-trisphosphate-induced calcium release, inhibits calcium pumps and has a use-dependent and slowly reversible action on store-operated calcium entry channels. [electronic resource]
Producer: 20040304Description: 97-108 p. digitalISSN:- 0143-4160
- Boron Compounds -- pharmacology
- Calcium Channels -- drug effects
- Calcium Signaling -- drug effects
- Calcium-Transporting ATPases -- antagonists & inhibitors
- Cell Membrane -- drug effects
- Cell Membrane Permeability -- drug effects
- Dose-Response Relationship, Drug
- Electric Stimulation
- HeLa Cells
- Humans
- Inositol 1,4,5-Trisphosphate -- antagonists & inhibitors
- Inositol 1,4,5-Trisphosphate Receptors
- Membrane Potentials -- drug effects
- Mitochondria -- drug effects
- Myocytes, Cardiac
- Receptors, Cytoplasmic and Nuclear -- antagonists & inhibitors
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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