T0070907, a selective ligand for peroxisome proliferator-activated receptor gamma, functions as an antagonist of biochemical and cellular activities. [electronic resource]
Producer: 20020702Description: 19649-57 p. digitalISSN:- 0021-9258
- 3T3 Cells
- Adipocytes -- cytology
- Allosteric Site
- Amino Acid Sequence
- Animals
- Anticarcinogenic Agents -- pharmacology
- Benzamides -- chemistry
- Bexarotene
- Cell Differentiation
- Cell Line
- Cysteine -- chemistry
- Dimerization
- Dose-Response Relationship, Drug
- Glutathione Transferase -- metabolism
- Humans
- Ligands
- Mice
- Molecular Sequence Data
- Mutation
- Peptides -- chemistry
- Plasmids -- metabolism
- Protein Binding
- Protein Conformation
- Protein Structure, Tertiary
- Pyridines -- chemistry
- Receptors, Cytoplasmic and Nuclear -- antagonists & inhibitors
- Receptors, Retinoic Acid -- metabolism
- Recombinant Fusion Proteins -- metabolism
- Retinoid X Receptors
- Spectrometry, Fluorescence
- Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
- Tetrahydronaphthalenes -- pharmacology
- Time Factors
- Transcription Factors -- antagonists & inhibitors
- Transcription, Genetic
- Transfection
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Publication Type: Journal Article
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