T0070907, a selective ligand for peroxisome proliferator-activated receptor gamma, functions as an antagonist of biochemical and cellular activities.

Lee, Gary

T0070907, a selective ligand for peroxisome proliferator-activated receptor gamma, functions as an antagonist of biochemical and cellular activities. [electronic resource] - The Journal of biological chemistry May 2002 - 19649-57 p. digital

Publication Type: Journal Article

0021-9258

10.1074/jbc.M200743200 doi


3T3 Cells
Adipocytes--cytology
Allosteric Site
Amino Acid Sequence
Animals
Anticarcinogenic Agents--pharmacology
Benzamides--chemistry
Bexarotene
Cell Differentiation
Cell Line
Cysteine--chemistry
Dimerization
Dose-Response Relationship, Drug
Glutathione Transferase--metabolism
Humans
Ligands
Mice
Molecular Sequence Data
Mutation
Peptides--chemistry
Plasmids--metabolism
Protein Binding
Protein Conformation
Protein Structure, Tertiary
Pyridines--chemistry
Receptors, Cytoplasmic and Nuclear--antagonists & inhibitors
Receptors, Retinoic Acid--metabolism
Recombinant Fusion Proteins--metabolism
Retinoid X Receptors
Spectrometry, Fluorescence
Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
Tetrahydronaphthalenes--pharmacology
Time Factors
Transcription Factors--antagonists & inhibitors
Transcription, Genetic
Transfection