Point mutations at multiple sites including highly conserved amino acids maintain activity, but render O6-alkylguanine-DNA alkyltransferase insensitive to O6-benzylguanine. [electronic resource]
Producer: 20010301Description: 519-26 p. digitalISSN:- 0264-6021
- Amino Acid Sequence
- Amino Acid Substitution -- genetics
- Antineoplastic Agents -- pharmacology
- Binding Sites
- Conserved Sequence -- genetics
- DNA Repair -- drug effects
- Drug Resistance -- genetics
- Escherichia coli
- Gene Library
- Guanine -- analogs & derivatives
- Humans
- Methylnitronitrosoguanidine -- pharmacology
- Molecular Sequence Data
- O(6)-Methylguanine-DNA Methyltransferase -- chemistry
- Point Mutation -- genetics
- Sequence Alignment
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Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
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