Complete Substrate Inhibition of Cytochrome P450 2C8 by AZD9496, an Oral Selective Estrogen Receptor Degrader. (Record no. 28549003)

MARC details
000 -LEADER
fixed length control field 01591 a2200421 4500
005 - DATE AND TIME OF LATEST TRANSACTION
control field 20250517223430.0
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION
fixed length control field 201812s 0 0 eng d
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER
International Standard Serial Number 1521-009X
024 7# - OTHER STANDARD IDENTIFIER
Standard number or code 10.1124/dmd.118.081539
Source of number or code doi
040 ## - CATALOGING SOURCE
Original cataloging agency NLM
Language of cataloging eng
Transcribing agency NLM
100 1# - MAIN ENTRY--PERSONAL NAME
Personal name Bapiro, Tashinga E
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE
Date of production, publication, distribution, manufacture, or copyright notice 20181211
245 00 - TITLE STATEMENT
Title Complete Substrate Inhibition of Cytochrome P450 2C8 by AZD9496, an Oral Selective Estrogen Receptor Degrader.
Medium [electronic resource]
260 ## - PUBLICATION, DISTRIBUTION, ETC.
Name of publisher, distributor, etc. Drug metabolism and disposition: the biological fate of chemicals
Date of publication, distribution, etc. 09 2018
300 ## - PHYSICAL DESCRIPTION
Extent 1268-1276 p.
Other physical details digital
500 ## - GENERAL NOTE
General note Publication Type: Journal Article; Research Support, Non-U.S. Gov't
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Administration, Oral
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cinnamates
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cytochrome P-450 CYP2C8
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cytochrome P-450 CYP2C8 Inhibitors
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Dose-Response Relationship, Drug
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Female
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Humans
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Indoles
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Male
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Microsomes, Liver
General subdivision drug effects
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Receptors, Estrogen
General subdivision antagonists & inhibitors
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Substrate Specificity
General subdivision drug effects
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Sykes, Andy
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Martin, Scott
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Davies, Michael
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Yates, James W T
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Hoch, Matthias
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Rollison, Helen E
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Jones, Barry
773 0# - HOST ITEM ENTRY
Title Drug metabolism and disposition: the biological fate of chemicals
Related parts vol. 46
-- no. 9
-- p. 1268-1276
856 40 - ELECTRONIC LOCATION AND ACCESS
Uniform Resource Identifier <a href="https://doi.org/10.1124/dmd.118.081539">https://doi.org/10.1124/dmd.118.081539</a>
Public note Available from publisher's website

No items available.