Novel Aryl Substituted Pyrazoles as Small Molecule Inhibitors of Cytochrome P450 CYP121A1: Synthesis and Antimycobacterial Evaluation. (Record no. 27835281)

MARC details
000 -LEADER
fixed length control field 01921 a2200505 4500
005 - DATE AND TIME OF LATEST TRANSACTION
control field 20250517185947.0
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION
fixed length control field 201904s 0 0 eng d
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER
International Standard Serial Number 1520-4804
024 7# - OTHER STANDARD IDENTIFIER
Standard number or code 10.1021/acs.jmedchem.7b01562
Source of number or code doi
040 ## - CATALOGING SOURCE
Original cataloging agency NLM
Language of cataloging eng
Transcribing agency NLM
100 1# - MAIN ENTRY--PERSONAL NAME
Personal name Taban, Ismail M
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE
Date of production, publication, distribution, manufacture, or copyright notice 20190401
245 00 - TITLE STATEMENT
Title Novel Aryl Substituted Pyrazoles as Small Molecule Inhibitors of Cytochrome P450 CYP121A1: Synthesis and Antimycobacterial Evaluation.
Medium [electronic resource]
260 ## - PUBLICATION, DISTRIBUTION, ETC.
Name of publisher, distributor, etc. Journal of medicinal chemistry
Date of publication, distribution, etc. 12 2017
300 ## - PHYSICAL DESCRIPTION
Extent 10257-10267 p.
Other physical details digital
500 ## - GENERAL NOTE
General note Publication Type: Journal Article; Research Support, Non-U.S. Gov't
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Antitubercular Agents
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Bacterial Proteins
General subdivision antagonists & inhibitors
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Binding Sites
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Crystallography, X-Ray
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cytochrome P-450 Enzyme Inhibitors
General subdivision chemical synthesis
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cytochrome P-450 Enzyme System
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Drug Evaluation, Preclinical
General subdivision methods
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Microbial Sensitivity Tests
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Molecular Docking Simulation
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Mycobacterium tuberculosis
General subdivision drug effects
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Pyrazoles
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Small Molecule Libraries
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Spectrophotometry, Ultraviolet
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Elshihawy, Hosam E A E
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Torun, Beyza
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Zucchini, Benedetta
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Williamson, Clare J
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Altuwairigi, Dania
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Ngu, Adeline S T
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name McLean, Kirsty J
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Levy, Colin W
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Sood, Sakshi
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Marino, Leonardo B
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Munro, Andrew W
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name de Carvalho, Luiz Pedro S
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Simons, Claire
773 0# - HOST ITEM ENTRY
Title Journal of medicinal chemistry
Related parts vol. 60
-- no. 24
-- p. 10257-10267
856 40 - ELECTRONIC LOCATION AND ACCESS
Uniform Resource Identifier <a href="https://doi.org/10.1021/acs.jmedchem.7b01562">https://doi.org/10.1021/acs.jmedchem.7b01562</a>
Public note Available from publisher's website

No items available.