Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors. (Record no. 24987418)

MARC details
000 -LEADER
fixed length control field 01673 a2200445 4500
005 - DATE AND TIME OF LATEST TRANSACTION
control field 20250517035520.0
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION
fixed length control field 201509s 0 0 eng d
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER
International Standard Serial Number 1520-4804
024 7# - OTHER STANDARD IDENTIFIER
Standard number or code 10.1021/acs.jmedchem.5b00613
Source of number or code doi
040 ## - CATALOGING SOURCE
Original cataloging agency NLM
Language of cataloging eng
Transcribing agency NLM
100 1# - MAIN ENTRY--PERSONAL NAME
Personal name Ran, Xu
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE
Date of production, publication, distribution, manufacture, or copyright notice 20150914
245 00 - TITLE STATEMENT
Title Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors.
Medium [electronic resource]
260 ## - PUBLICATION, DISTRIBUTION, ETC.
Name of publisher, distributor, etc. Journal of medicinal chemistry
Date of publication, distribution, etc. Jun 2015
300 ## - PHYSICAL DESCRIPTION
Extent 4927-39 p.
Other physical details digital
500 ## - GENERAL NOTE
General note Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Antineoplastic Agents
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Carbolines
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cell Cycle Proteins
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cell Line, Tumor
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Crystallography, X-Ray
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Humans
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Leukemia
General subdivision drug therapy
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Molecular Docking Simulation
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Nuclear Proteins
General subdivision antagonists & inhibitors
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Protein Serine-Threonine Kinases
General subdivision antagonists & inhibitors
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element RNA-Binding Proteins
General subdivision antagonists & inhibitors
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Transcription Factors
General subdivision antagonists & inhibitors
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Zhao, Yujun
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Liu, Liu
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Bai, Longchuan
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Yang, Chao-Yie
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Zhou, Bing
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Meagher, Jennifer L
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Chinnaswamy, Krishnapriya
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Stuckey, Jeanne A
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Wang, Shaomeng
773 0# - HOST ITEM ENTRY
Title Journal of medicinal chemistry
Related parts vol. 58
-- no. 12
-- p. 4927-39
856 40 - ELECTRONIC LOCATION AND ACCESS
Uniform Resource Identifier <a href="https://doi.org/10.1021/acs.jmedchem.5b00613">https://doi.org/10.1021/acs.jmedchem.5b00613</a>
Public note Available from publisher's website

No items available.