Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors.
Ran, Xu
Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors. [electronic resource] - Journal of medicinal chemistry Jun 2015 - 4927-39 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4804
10.1021/acs.jmedchem.5b00613 doi
Antineoplastic Agents--chemistry
Carbolines--chemistry
Cell Cycle Proteins
Cell Line, Tumor
Crystallography, X-Ray
Humans
Leukemia--drug therapy
Molecular Docking Simulation
Nuclear Proteins--antagonists & inhibitors
Protein Serine-Threonine Kinases--antagonists & inhibitors
RNA-Binding Proteins--antagonists & inhibitors
Transcription Factors--antagonists & inhibitors
Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors. [electronic resource] - Journal of medicinal chemistry Jun 2015 - 4927-39 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4804
10.1021/acs.jmedchem.5b00613 doi
Antineoplastic Agents--chemistry
Carbolines--chemistry
Cell Cycle Proteins
Cell Line, Tumor
Crystallography, X-Ray
Humans
Leukemia--drug therapy
Molecular Docking Simulation
Nuclear Proteins--antagonists & inhibitors
Protein Serine-Threonine Kinases--antagonists & inhibitors
RNA-Binding Proteins--antagonists & inhibitors
Transcription Factors--antagonists & inhibitors