2-(3-Oxo-1,3-diphenylpropyl)malonic acids as potent allosteric ligands of the PIF pocket of phosphoinositide-dependent kinase-1: development and prodrug concept. (Record no. 22220409)
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fixed length control field | 01856 a2200505 4500 |
005 - DATE AND TIME OF LATEST TRANSACTION | |
control field | 20250516120158.0 |
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
fixed length control field | 201302s 0 0 eng d |
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
International Standard Serial Number | 1520-4804 |
024 7# - OTHER STANDARD IDENTIFIER | |
Standard number or code | 10.1021/jm3010477 |
Source of number or code | doi |
040 ## - CATALOGING SOURCE | |
Original cataloging agency | NLM |
Language of cataloging | eng |
Transcribing agency | NLM |
100 1# - MAIN ENTRY--PERSONAL NAME | |
Personal name | Wilhelm, Adriana |
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
Date of production, publication, distribution, manufacture, or copyright notice | 20130205 |
245 00 - TITLE STATEMENT | |
Title | 2-(3-Oxo-1,3-diphenylpropyl)malonic acids as potent allosteric ligands of the PIF pocket of phosphoinositide-dependent kinase-1: development and prodrug concept. |
Medium | [electronic resource] |
260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
Name of publisher, distributor, etc. | Journal of medicinal chemistry |
Date of publication, distribution, etc. | Nov 2012 |
300 ## - PHYSICAL DESCRIPTION | |
Extent | 9817-30 p. |
Other physical details | digital |
500 ## - GENERAL NOTE | |
General note | Publication Type: Journal Article; Research Support, Non-U.S. Gov't |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Allosteric Site |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Binding Sites |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | DNA Helicases |
General subdivision | antagonists & inhibitors |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Drug Design |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Enzyme Activation |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Humans |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Immunoblotting |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Malonates |
General subdivision | chemical synthesis |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Models, Molecular |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Molecular Structure |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Muscle Cells |
General subdivision | drug effects |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Prodrugs |
General subdivision | chemical synthesis |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Protein Binding |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Protein Kinase Inhibitors |
General subdivision | chemical synthesis |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Protein Serine-Threonine Kinases |
General subdivision | antagonists & inhibitors |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Pyruvate Dehydrogenase Acetyl-Transferring Kinase |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Structure-Activity Relationship |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Lopez-Garcia, Laura A |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Busschots, Katrien |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Fröhner, Wolfgang |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Maurer, Frauke |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Boettcher, Stefan |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Zhang, Hua |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Schulze, Jörg O |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Biondi, Ricardo M |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Engel, Matthias |
773 0# - HOST ITEM ENTRY | |
Title | Journal of medicinal chemistry |
Related parts | vol. 55 |
-- | no. 22 |
-- | p. 9817-30 |
856 40 - ELECTRONIC LOCATION AND ACCESS | |
Uniform Resource Identifier | <a href="https://doi.org/10.1021/jm3010477">https://doi.org/10.1021/jm3010477</a> |
Public note | Available from publisher's website |
No items available.