Synthesis and structure-activity relationships of 4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1-hi]indoles: novel PDE4 inhibitors. (Record no. 10591570)

MARC details
000 -LEADER
fixed length control field 01870 a2200565 4500
005 - DATE AND TIME OF LATEST TRANSACTION
control field 20250513201532.0
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION
fixed length control field 200002s 0 0 eng d
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER
International Standard Serial Number 0960-894X
024 7# - OTHER STANDARD IDENTIFIER
Standard number or code 10.1016/s0960-894x(99)00573-9
Source of number or code doi
040 ## - CATALOGING SOURCE
Original cataloging agency NLM
Language of cataloging eng
Transcribing agency NLM
100 1# - MAIN ENTRY--PERSONAL NAME
Personal name Pascal, Y
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE
Date of production, publication, distribution, manufacture, or copyright notice 20000228
245 00 - TITLE STATEMENT
Title Synthesis and structure-activity relationships of 4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1-hi]indoles: novel PDE4 inhibitors.
Medium [electronic resource]
260 ## - PUBLICATION, DISTRIBUTION, ETC.
Name of publisher, distributor, etc. Bioorganic & medicinal chemistry letters
Date of publication, distribution, etc. Jan 2000
300 ## - PHYSICAL DESCRIPTION
Extent 35-8 p.
Other physical details digital
500 ## - GENERAL NOTE
General note Publication Type: Journal Article
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element 3',5'-Cyclic-AMP Phosphodiesterases
General subdivision antagonists & inhibitors
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Animals
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Benzodiazepines
General subdivision chemical synthesis
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Binding Sites
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Cyclic Nucleotide Phosphodiesterases, Type 4
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Dogs
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Guinea Pigs
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Humans
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Indoles
General subdivision chemical synthesis
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Inhibitory Concentration 50
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Phosphodiesterase Inhibitors
General subdivision chemical synthesis
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Rats
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Rats, Inbred BN
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Rats, Wistar
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Rolipram
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Stereoisomerism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Structure-Activity Relationship
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Substrate Specificity
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element U937 Cells
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Andrianjara, C R
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Auclair, E
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Avenel, N
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Bertin, B
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Calvet, A
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Féru, F
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Lardon, S
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Moodley, I
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Ouagued, M
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Payne, A
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Pruniaux, M P
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Szilagyi, C
773 0# - HOST ITEM ENTRY
Title Bioorganic & medicinal chemistry letters
Related parts vol. 10
-- no. 1
-- p. 35-8
856 40 - ELECTRONIC LOCATION AND ACCESS
Uniform Resource Identifier <a href="https://doi.org/10.1016/s0960-894x(99)00573-9">https://doi.org/10.1016/s0960-894x(99)00573-9</a>
Public note Available from publisher's website

No items available.