Co-targeting bromodomain and extra-terminal proteins and MCL1 induces synergistic cell death in melanoma.

Tseng, Hsin-Yi

Co-targeting bromodomain and extra-terminal proteins and MCL1 induces synergistic cell death in melanoma. [electronic resource] - International journal of cancer 10 2020 - 2176-2189 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1097-0215

10.1002/ijc.33000 doi


Animals
Antineoplastic Agents--pharmacology
Apoptosis--drug effects
Apoptosis Regulatory Proteins--metabolism
Cell Death--drug effects
Cell Line, Tumor
Down-Regulation--drug effects
Drug Resistance, Neoplasm--drug effects
Drug Synergism
Humans
Male
Melanoma--drug therapy
Mice
Mice, Inbred NOD
Mice, SCID
Myeloid Cell Leukemia Sequence 1 Protein--metabolism
Proteins--metabolism
Pyrimidines--pharmacology
Thiophenes--pharmacology
Up-Regulation--drug effects