Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors.

Kufareva, Irina

Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors. [electronic resource] - Scientific reports 11 2019 - 15893 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

2045-2322

10.1038/s41598-019-52141-5 doi


Adenosine Triphosphate--metabolism
Binding Sites
Casein Kinase II--antagonists & inhibitors
Catalytic Domain
Cell Line, Tumor
Cell Movement--drug effects
Cell Proliferation--drug effects
Crystallography, X-Ray
Holoenzymes--chemistry
Humans
Kinetics
Molecular Docking Simulation
Peptides--chemistry
Phosphorylation
Protein Kinase Inhibitors--chemistry
Protein Subunits--antagonists & inhibitors
Substrate Specificity
Surface Plasmon Resonance