Structure Overhaul Affords a Potent Purine PI3Kδ Inhibitor with Improved Tolerability.
Methot, Joey L
Structure Overhaul Affords a Potent Purine PI3Kδ Inhibitor with Improved Tolerability. [electronic resource] - Journal of medicinal chemistry 05 2019 - 4370-4382 p. digital
Publication Type: Journal Article
1520-4804
10.1021/acs.jmedchem.8b01818 doi
Animals
Class Ia Phosphatidylinositol 3-Kinase--metabolism
Dogs
Drug Design
HeLa Cells
Humans
Male
Protein Kinase Inhibitors--chemical synthesis
Purines--chemical synthesis
Pyrrolidines--chemical synthesis
Rats, Wistar
Structure Overhaul Affords a Potent Purine PI3Kδ Inhibitor with Improved Tolerability. [electronic resource] - Journal of medicinal chemistry 05 2019 - 4370-4382 p. digital
Publication Type: Journal Article
1520-4804
10.1021/acs.jmedchem.8b01818 doi
Animals
Class Ia Phosphatidylinositol 3-Kinase--metabolism
Dogs
Drug Design
HeLa Cells
Humans
Male
Protein Kinase Inhibitors--chemical synthesis
Purines--chemical synthesis
Pyrrolidines--chemical synthesis
Rats, Wistar