SKLB188 inhibits the growth of head and neck squamous cell carcinoma by suppressing EGFR signalling.

Barzegar, Mansoureh

SKLB188 inhibits the growth of head and neck squamous cell carcinoma by suppressing EGFR signalling. [electronic resource] - British journal of cancer Oct 2017 - 1154-1163 p. digital

Publication Type: Journal Article

1532-1827

10.1038/bjc.2017.298 doi


Animals
Apoptosis--drug effects
Blotting, Western
Carcinoma, Squamous Cell--metabolism
Cell Proliferation--drug effects
Cyclin A--drug effects
Cyclin D1--drug effects
Cyclin-Dependent Kinase 2--drug effects
Cyclin-Dependent Kinase 4--drug effects
Cyclin-Dependent Kinase Inhibitor p21--drug effects
Cyclin-Dependent Kinase Inhibitor p27--drug effects
Down-Regulation
ErbB Receptors--antagonists & inhibitors
G1 Phase Cell Cycle Checkpoints--drug effects
Head and Neck Neoplasms--metabolism
Humans
Immunohistochemistry
In Situ Nick-End Labeling
In Vitro Techniques
Mice
Mice, Nude
Molecular Docking Simulation
Purines--pharmacology
Signal Transduction
Squamous Cell Carcinoma of Head and Neck
Up-Regulation
Xenograft Model Antitumor Assays
cdc25 Phosphatases--drug effects