Oxidized 5-aminosalicylic acid activates Nrf2-HO-1 pathway by covalently binding to Keap1: Implication in anti-inflammatory actions of 5-aminosalicylic acid.
Kang, Sookjin
Oxidized 5-aminosalicylic acid activates Nrf2-HO-1 pathway by covalently binding to Keap1: Implication in anti-inflammatory actions of 5-aminosalicylic acid. [electronic resource] - Free radical biology & medicine 07 2017 - 715-724 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-4596
10.1016/j.freeradbiomed.2017.04.366 doi
Animals
Anti-Inflammatory Agents--therapeutic use
Colonic Neoplasms--drug therapy
HCT116 Cells
Heme Oxygenase-1--metabolism
Humans
Hypochlorous Acid--metabolism
Inflammation--drug therapy
Inflammatory Bowel Diseases--drug therapy
Kelch-Like ECH-Associated Protein 1--metabolism
Male
Mesalamine--therapeutic use
NF-E2-Related Factor 2--metabolism
Oxidation-Reduction
Protein Binding
Rats
Rats, Sprague-Dawley
Oxidized 5-aminosalicylic acid activates Nrf2-HO-1 pathway by covalently binding to Keap1: Implication in anti-inflammatory actions of 5-aminosalicylic acid. [electronic resource] - Free radical biology & medicine 07 2017 - 715-724 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-4596
10.1016/j.freeradbiomed.2017.04.366 doi
Animals
Anti-Inflammatory Agents--therapeutic use
Colonic Neoplasms--drug therapy
HCT116 Cells
Heme Oxygenase-1--metabolism
Humans
Hypochlorous Acid--metabolism
Inflammation--drug therapy
Inflammatory Bowel Diseases--drug therapy
Kelch-Like ECH-Associated Protein 1--metabolism
Male
Mesalamine--therapeutic use
NF-E2-Related Factor 2--metabolism
Oxidation-Reduction
Protein Binding
Rats
Rats, Sprague-Dawley