Inhibitory studies of mexiletine and dextromethorphan oxidation in human liver microsomes.

Broly, F

Inhibitory studies of mexiletine and dextromethorphan oxidation in human liver microsomes. [electronic resource] - Biochemical pharmacology Mar 1990 - 1045-53 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0006-2952

10.1016/0006-2952(90)90283-q doi


Binding, Competitive
Cytochrome P-450 CYP2D6
Cytochrome P-450 Enzyme Inhibitors
Dealkylation
Dextromethorphan--metabolism
Drug Interactions
Humans
Hydroxylation
Immune Sera--pharmacology
In Vitro Techniques
Levorphanol--analogs & derivatives
Mexiletine--metabolism
Microsomes, Liver--metabolism
Mixed Function Oxygenases--antagonists & inhibitors
Oxidation-Reduction