Sarcophine-diol inhibits expression of COX-2, inhibits activity of cPLA2, enhances degradation of PLA2 and PLC(γ)1 and inhibits cell membrane permeability in mouse melanoma B16F10 cells.
Szymanski, Pawel T
Sarcophine-diol inhibits expression of COX-2, inhibits activity of cPLA2, enhances degradation of PLA2 and PLC(γ)1 and inhibits cell membrane permeability in mouse melanoma B16F10 cells. [electronic resource] - Marine drugs Oct 2012 - 2166-2180 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1660-3397
10.3390/md10102166 doi
Animals
Anthozoa--chemistry
Antineoplastic Agents--pharmacology
Cell Line, Tumor
Cell Membrane Permeability--drug effects
Cell Proliferation
Cyclooxygenase 2--genetics
Cyclooxygenase 2 Inhibitors--pharmacology
Diterpenes--chemistry
Gene Expression Regulation, Enzymologic
Melanoma--metabolism
Mice
Molecular Structure
Phospholipase C gamma--genetics
Phospholipases A2, Cytosolic--antagonists & inhibitors
Sarcophine-diol inhibits expression of COX-2, inhibits activity of cPLA2, enhances degradation of PLA2 and PLC(γ)1 and inhibits cell membrane permeability in mouse melanoma B16F10 cells. [electronic resource] - Marine drugs Oct 2012 - 2166-2180 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1660-3397
10.3390/md10102166 doi
Animals
Anthozoa--chemistry
Antineoplastic Agents--pharmacology
Cell Line, Tumor
Cell Membrane Permeability--drug effects
Cell Proliferation
Cyclooxygenase 2--genetics
Cyclooxygenase 2 Inhibitors--pharmacology
Diterpenes--chemistry
Gene Expression Regulation, Enzymologic
Melanoma--metabolism
Mice
Molecular Structure
Phospholipase C gamma--genetics
Phospholipases A2, Cytosolic--antagonists & inhibitors