Electron density guided fragment-based drug design--a lead generation example.

Abad, Marta C

Electron density guided fragment-based drug design--a lead generation example. [electronic resource] - Methods in enzymology 2011 - 487-508 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.

1557-7988

10.1016/B978-0-12-381274-2.00019-4 doi


Adenosine Triphosphate--metabolism
Adenylyl Imidodiphosphate--metabolism
Catalytic Domain--drug effects
Crystallography, X-Ray
Drug Design
Drug Discovery
Drug Evaluation, Preclinical--methods
Electrons
Enzyme Inhibitors--chemistry
Fructokinases--antagonists & inhibitors
Fructose--metabolism
Hydrogen Bonding
Models, Molecular
Protein Binding
Small Molecule Libraries
Sulfates--chemistry