Fragment-based drug discovery applied to Hsp90. Discovery of two lead series with high ligand efficiency.

Murray, Christopher W

Fragment-based drug discovery applied to Hsp90. Discovery of two lead series with high ligand efficiency. [electronic resource] - Journal of medicinal chemistry Aug 2010 - 5942-55 p. digital

Publication Type: Journal Article

1520-4804

10.1021/jm100059d doi


Aminopyridines--chemical synthesis
Antineoplastic Agents--chemistry
Crystallography, X-Ray
Databases, Factual
Drug Design
HSP90 Heat-Shock Proteins--antagonists & inhibitors
Ligands
Magnetic Resonance Spectroscopy
Models, Molecular
Phenols--chemical synthesis
Protein Binding
Protein Structure, Tertiary
Resorcinols--chemical synthesis
Structure-Activity Relationship