Activation of alpha4* nAChRs is necessary and sufficient for varenicline-induced reduction of alcohol consumption.
Hendrickson, Linzy M
Activation of alpha4* nAChRs is necessary and sufficient for varenicline-induced reduction of alcohol consumption. [electronic resource] - The Journal of neuroscience : the official journal of the Society for Neuroscience Jul 2010 - 10169-76 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1529-2401
10.1523/JNEUROSCI.2601-10.2010 doi
Alanine--genetics
Alcohol Drinking--drug therapy
Analysis of Variance
Animals
Benzazepines--therapeutic use
Central Nervous System Depressants--administration & dosage
Disease Models, Animal
Dopamine--metabolism
Dose-Response Relationship, Drug
Drinking Behavior--drug effects
Drug Combinations
Ethanol--administration & dosage
Gene Expression Regulation--drug effects
Leucine--genetics
Male
Mice
Mice, Inbred C57BL
Mice, Transgenic
Mutation--genetics
Neurons--drug effects
Nicotinic Agonists--therapeutic use
Proto-Oncogene Proteins c-fos--metabolism
Quinoxalines--therapeutic use
Receptors, Nicotinic--deficiency
Tyrosine 3-Monooxygenase--metabolism
Varenicline
Ventral Tegmental Area--cytology
Activation of alpha4* nAChRs is necessary and sufficient for varenicline-induced reduction of alcohol consumption. [electronic resource] - The Journal of neuroscience : the official journal of the Society for Neuroscience Jul 2010 - 10169-76 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1529-2401
10.1523/JNEUROSCI.2601-10.2010 doi
Alanine--genetics
Alcohol Drinking--drug therapy
Analysis of Variance
Animals
Benzazepines--therapeutic use
Central Nervous System Depressants--administration & dosage
Disease Models, Animal
Dopamine--metabolism
Dose-Response Relationship, Drug
Drinking Behavior--drug effects
Drug Combinations
Ethanol--administration & dosage
Gene Expression Regulation--drug effects
Leucine--genetics
Male
Mice
Mice, Inbred C57BL
Mice, Transgenic
Mutation--genetics
Neurons--drug effects
Nicotinic Agonists--therapeutic use
Proto-Oncogene Proteins c-fos--metabolism
Quinoxalines--therapeutic use
Receptors, Nicotinic--deficiency
Tyrosine 3-Monooxygenase--metabolism
Varenicline
Ventral Tegmental Area--cytology