Amplification of EGFR T790M causes resistance to an irreversible EGFR inhibitor.

Ercan, D

Amplification of EGFR T790M causes resistance to an irreversible EGFR inhibitor. [electronic resource] - Oncogene Apr 2010 - 2346-56 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1476-5594

10.1038/onc.2009.526 doi


Carcinoma, Non-Small-Cell Lung--drug therapy
Cell Line, Tumor
Drug Resistance, Neoplasm
ErbB Receptors--antagonists & inhibitors
Gefitinib
Gene Amplification
Humans
Lung Neoplasms--drug therapy
Phosphorylation
Protein Kinase Inhibitors--pharmacology
Quinazolines--pharmacology
Quinazolinones--pharmacology