The marine phycotoxin gymnodimine targets muscular and neuronal nicotinic acetylcholine receptor subtypes with high affinity.

Kharrat, Riadh

The marine phycotoxin gymnodimine targets muscular and neuronal nicotinic acetylcholine receptor subtypes with high affinity. [electronic resource] - Journal of neurochemistry Nov 2008 - 952-63 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1471-4159

10.1111/j.1471-4159.2008.05677.x doi


Acetylcholine--pharmacology
Animals
Behavior, Animal--drug effects
Bivalvia--chemistry
Bungarotoxins--metabolism
Cells, Cultured
Chromatography, High Pressure Liquid--methods
Dose-Response Relationship, Drug
Drug Interactions
Electric Stimulation--methods
Gene Expression--drug effects
Heterocyclic Compounds, 3-Ring--analysis
Humans
Hydrocarbons, Cyclic--analysis
Imines--analysis
Male
Membrane Potentials--drug effects
Mice
Mice, Inbred C57BL
Muscle Cells--drug effects
Neuromuscular Junction--drug effects
Oocytes
Patch-Clamp Techniques
Protein Binding--drug effects
Receptors, Nicotinic--metabolism
Synaptic Transmission--drug effects
Xenopus laevis
alpha7 Nicotinic Acetylcholine Receptor