Effects of KP-496, a novel dual antagonist at the cysteinyl leukotriene receptor 1 and the thromboxane A(2) receptor, on airway obstruction in guinea pigs.

Ishimura, M

Effects of KP-496, a novel dual antagonist at the cysteinyl leukotriene receptor 1 and the thromboxane A(2) receptor, on airway obstruction in guinea pigs. [electronic resource] - British journal of pharmacology Feb 2008 - 669-75 p. digital

Publication Type: Comparative Study; Journal Article

0007-1188

10.1038/sj.bjp.0707602 doi


15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid
Acetates--pharmacology
Administration, Inhalation
Administration, Oral
Airway Obstruction--chemically induced
Animals
Anti-Asthmatic Agents--administration & dosage
Benzoates--administration & dosage
Benzoquinones--pharmacology
Bronchoconstriction--drug effects
Cyclopropanes
Disease Models, Animal
Dose-Response Relationship, Drug
Drug Therapy, Combination
Guinea Pigs
Heptanoic Acids--pharmacology
Leukotriene Antagonists--administration & dosage
Leukotriene D4
Lung--drug effects
Male
Membrane Proteins--antagonists & inhibitors
Ovalbumin
Prostaglandin Antagonists--administration & dosage
Quinolines--pharmacology
Receptors, Leukotriene--metabolism
Receptors, Thromboxane A2, Prostaglandin H2--antagonists & inhibitors
Respiratory Hypersensitivity--immunology
Sulfides
Thiazoles--administration & dosage
Time Factors