Pharmacological profile of CR3465, a new leukotriene CysLT1 receptor antagonist with broad anti-inflammatory activity.

Ferrari, Flora

Pharmacological profile of CR3465, a new leukotriene CysLT1 receptor antagonist with broad anti-inflammatory activity. [electronic resource] - European journal of pharmacology Nov 2004 - 223-33 p. digital

Publication Type: Journal Article

0014-2999

10.1016/j.ejphar.2004.10.010 doi


3',5'-Cyclic-AMP Phosphodiesterases--antagonists & inhibitors
Animals
Anti-Inflammatory Agents
Bronchoalveolar Lavage Fluid--cytology
Bronchoconstriction--drug effects
Cell Degranulation--drug effects
Cyclic Nucleotide Phosphodiesterases, Type 3
Cyclic Nucleotide Phosphodiesterases, Type 4
Guinea Pigs
Histamine--pharmacology
Histamine Antagonists--pharmacology
Humans
In Vitro Techniques
Leukotriene D4--antagonists & inhibitors
Membrane Proteins--antagonists & inhibitors
N-Formylmethionine Leucyl-Phenylalanine--pharmacology
Neutrophils--drug effects
Parasympatholytics--pharmacology
Peroxidase--metabolism
Phosphodiesterase Inhibitors--pharmacology
Quinolines--pharmacology
Radioligand Assay
Rats
Receptors, Leukotriene
Tumor Necrosis Factor-alpha--metabolism
Tyrosine--analogs & derivatives