A novel mutant allele of the CYP2A6 gene (CYP2A6*11 ) found in a cancer patient who showed poor metabolic phenotype towards tegafur.
Daigo, Satoshi
A novel mutant allele of the CYP2A6 gene (CYP2A6*11 ) found in a cancer patient who showed poor metabolic phenotype towards tegafur. [electronic resource] - Pharmacogenetics Jun 2002 - 299-306 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0960-314X
10.1097/00008571-200206000-00005 doi
Administration, Oral
Antimetabolites, Antineoplastic--administration & dosage
Area Under Curve
Aryl Hydrocarbon Hydroxylases--genetics
Coumarins--metabolism
Cytochrome P-450 CYP2A6
DNA Primers--chemistry
DNA, Neoplasm--blood
Drug Combinations
Escherichia coli
Genotype
Humans
Kinetics
Middle Aged
Mixed Function Oxygenases--genetics
Mutagenesis, Site-Directed
Oxonic Acid--administration & dosage
Polymerase Chain Reaction
Polymorphism, Genetic
Pyridines--administration & dosage
Recombinant Proteins--isolation & purification
Stomach Neoplasms--enzymology
Tegafur--administration & dosage
Transfection
A novel mutant allele of the CYP2A6 gene (CYP2A6*11 ) found in a cancer patient who showed poor metabolic phenotype towards tegafur. [electronic resource] - Pharmacogenetics Jun 2002 - 299-306 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0960-314X
10.1097/00008571-200206000-00005 doi
Administration, Oral
Antimetabolites, Antineoplastic--administration & dosage
Area Under Curve
Aryl Hydrocarbon Hydroxylases--genetics
Coumarins--metabolism
Cytochrome P-450 CYP2A6
DNA Primers--chemistry
DNA, Neoplasm--blood
Drug Combinations
Escherichia coli
Genotype
Humans
Kinetics
Middle Aged
Mixed Function Oxygenases--genetics
Mutagenesis, Site-Directed
Oxonic Acid--administration & dosage
Polymerase Chain Reaction
Polymorphism, Genetic
Pyridines--administration & dosage
Recombinant Proteins--isolation & purification
Stomach Neoplasms--enzymology
Tegafur--administration & dosage
Transfection