Inhibition of all-TRANS-retinoic acid metabolism by R116010 induces antitumour activity.

Van Heusden, J

Inhibition of all-TRANS-retinoic acid metabolism by R116010 induces antitumour activity. [electronic resource] - British journal of cancer Feb 2002 - 605-11 p. digital

Publication Type: Comparative Study; Journal Article

0007-0920

10.1038/sj.bjc.6600056 doi


Animals
Antineoplastic Agents--pharmacology
Benzothiazoles
Breast Neoplasms--metabolism
Cell Division--drug effects
Chromatography, High Pressure Liquid
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--genetics
Dose-Response Relationship, Drug
Female
Humans
Imidazoles--pharmacology
Mammary Neoplasms, Experimental--metabolism
Mice
Mice, Inbred Strains
Mixed Function Oxygenases--antagonists & inhibitors
Retinoic Acid 4-Hydroxylase
Reverse Transcriptase Polymerase Chain Reaction
Thiazoles--pharmacology
Tretinoin--metabolism
Tumor Cells, Cultured--drug effects