Isoflurane increases the apparent agonist affinity of the nicotinic acetylcholine receptor by reducing the microscopic agonist dissociation constant.

Raines, D E

Isoflurane increases the apparent agonist affinity of the nicotinic acetylcholine receptor by reducing the microscopic agonist dissociation constant. [electronic resource] - Anesthesiology Mar 2000 - 775-85 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0003-3022

10.1097/00000542-200003000-00021 doi


Algorithms
Anesthetics, Inhalation--pharmacology
Animals
Choline--analogs & derivatives
Cholinergic Agents--metabolism
Dansyl Compounds
Fluorescent Dyes
In Vitro Techniques
Ion Channel Gating--drug effects
Isoflurane--pharmacology
Kinetics
Membranes--drug effects
Nicotinic Agonists--pharmacology
Quaternary Ammonium Compounds
Receptors, Nicotinic--drug effects
Spectrometry, Fluorescence
Torpedo